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Soares, Daniela Fernandes Ramos; Groll, Andrea Von; Ramis, Ivy Bastos; Coelho, Tatiane Silveira; Flach, Juliana; Silva, Pedro Eduardo Almeida da
(2008)
A tuberculose (TB) é uma doença infecciosa com uma incidência mundial estimada de 8,8
milhões de casos. Considerando o aumento no número de casos por cepas
multidrogarresistente (MDR-TB) e o reduzido arsenal terapêutico, ...
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Volcão, Lisiane Martins; Coelho, Tatiane Silveira; Vàsquez, Alváro; Cerdeiras, Maria Pia; Silva, Pedro Eduardo Almeida da; Silva Júnior, Flávio Manoel Rodrigues da; Soares, Daniela Fernandes Ramos
(2016)
Justificativa e Objetivos: O estudo objetivou a avaliação da atividade antibacteriana de extratos brutos e frações
de Ibicella lutea, na inibição do crescimento de Staphylococcus aureus, avaliando a combinação destes ...
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Coelho, Tatiane Silveira; Machado, Diana; Couto, Isabel; Maschmann, Raquel Abreu; Soares, Daniela Fernandes Ramos; Groll, Andrea Von; Rossetti, Maria Lucia Rosa; Silva, Pedro Almeida da; Viveiros, Miguel
(2015)
Drug resistant tuberculosis continues to increase and new approaches for its treatment
are necessary. The identification of M. tuberculosis clinical isolates presenting efflux
as part of their resistant phenotype has a ...
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Coelho, Tatiane Silveira; Cantos, Jéssica Borges; Bispo, Marcelle; Gonçalves, Raoni Schroeder Borges; Lima, Camilo Henrique da Silva; Silva, Pedro Eduardo Almeida da; Souza, Marcus Vinícius Nora de
(2012)
A series of twenty-three N-acylhydrazones
derived from isoniazid (INH 1-23) have been
evaluated for their in vitro antibacterial activity against INH- susceptible strain of M. tuberculosis (RG500) and three INH-resistant ...
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Carneiro, Paula Fernandes; Pinto, Maria do Carmo Freire Ribeiro; Coelho, Tatiane Silveira; Cavalcanti, Bruno Coêlho; Pessoa, Cláudia; Simone, Carlos Alberto de; Nunes, Isabelle Karine da Costa; Oliveira, Nathália Milanez de; Almeida, Renata Gomes de; Pinto, Antonio Ventura; Moura, Kelly Cristina Gallan de; Pedro, Eduardo Almeida da; Silva Júnior, Eufrânio Nunes da
(2011)
Several quinonoid and phenazine compounds were synthesized in moderate to high yields and showed activity against H37Rv, rifampicin and isoniazid-resistance strains of Mycobacterium tuberculosis. The cytotoxity of the ...
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Rodrigues, Marieli Oliveira; Cantos, Jéssica Borges; D'Oca, Caroline Da Ros Montes; Soares, Karina Lotz; Coelho, Tatiane Silveira; Piovesan, Luciana Almeida; Russowsky, Dennis; Silva, Pedro Eduardo Almeida da; D'Oca, Marcelo Gonçalves Montes
(Elsevier, 2013)
This work describes the synthesis of a series of fatty acid hydrazide derivatives of isoniazid (INH). The compounds were tested against Mycobacterium tuberculosis H37Rv (ATCC 27294) as well as INH-resistant (ATCC 35822 and ...
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D'Oca, Caroline Da Ros Montes; Coelho, Tatiane Silveira; Marinho, Tamara Germani; Hack, Carolina Rosa Lopes; Duarte, Rodrigo da Costa; Silva, Pedro Eduardo Almeida da; D'Oca, Marcelo Gonçalves Montes
(2010)
This work reports the synthesis of new fatty acid amides from C16:0, 18:0, 18:1, 18:1 (OH), and 18:2 fatty acids families with cyclic and acyclic amines and demonstrate for the first time the activity of these compounds ...
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Silva, Pedro Eduardo Almeida da; Soares, Daniela Fernandes Ramos; Bonacorso, Helio Gauze; Iglesia, Agustina de la; Oliveira, Marli Redin; Coelho, Tatiane Silveira; Navarini, Jussara; Morbidoni, Hector; Zanatta, Nilo; Martins, Marcos Antonio Pinto
(2008)
A series of 3-substituted 5-hydroxy-5-trifluoro[chloro]methyl-1H-1-isonicotinoyl-4,5-dihydropyrazoles (2a–i) were synthesised by the cyclocondensation reaction of 4-methoxy-1,1,1-trifluoro[chloro]-4 (substituted)-alk-3-en-2-ones ...
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Duarte, Aline Castellar; Coelho, Tatiane Silveira; Silva, Pedro Eduardo Almeida da; Soares, Daniela Fernandes Ramos; Lourenço, Maria Cristina da Silva; Lage, Celso Luiz Salgueiro; Julião, Lisieux de Santana; Barbosa, Ymira Albuquerque Gálico; Leitão, Suzana Guimarães
(2011)
Tuberculosis (TB), caused by Mycobacterium tuberculosis, is the world’s number one killer among infectious diseases. The search for new natural products that can act as drugs against TB has received increased attention ...